【Batch】Gallium-68 radiolabeling reaction of DOTA derivatives (Chelate reaction)1 【バッチ】PET核種68Gaを用いた配位子DOTAへのキレート反応1
J. Label. Compd. Radiopharm., 62, 132-138 (2019).

Outline

J. Label. Compd. Radiopharm., 62, 132-138 (2019).
DOI: 10.1016/j.tetlet.2022.154010

“Efficient gallium-68 radiolabeling reaction of DOTA derivatives using a resonant-type microwave reactor”

Yusuke Yagi 1 , Yoichi Shimizu 2 , Kenji Arimitsu 1 , Yuji Nakamoto 3 , Takahiro Higuchi 4 , Kaori Togashi 3 , Hiroyuki Kimura 1

1 Department of Analytical and Bioinorganic Chemistry, Division of Analytical and Physical Sciences, Kyoto Pharmaceutical University, 5 Nakauchi-cho, Misasagi, Yamashina-ku, Kyoto 607-8414, Japan
2 Department of Radiology, Kyoto University Hospital, Kyoto, Japan
3 Department of Diagnostic Imaging and Nuclear Medicine, Kyoto University Graduate School of Medicine, Kyoto, Japan
4 Department of Nuclear Medicine/Comprehensive Heart Failure Center, University Hospital Würzburg, Würzburg, Germany

Equipment information Reactor size: batch-type microwave reactor, Maximum power: 10 W (SAIDA FDS INC.)

概要

実験結果提供:
京都薬科大学 屋木 祐亮先生、有光 健治先生、木村 寛之先生
京都大学医学部付属病院 志水 陽一先生
京都大学医学部 中本 裕士先生、富樫 かおり先生
ヴェルツブルク大学、岡山大学 樋口 隆弘先生

装置情報:バッチ型マイクロ波装置、10 W

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